Drugs that cause Gynaecomastia
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LIST 1
Drugs that can cause gynaecomastia
Anti-arrythmic drugs
Digoxin
Anti-psychotic or neuroleptic drugs
Amisulpiride
Aripiprazole
Benperidlo
Chlorpromazine
Clozapine
Flupentixol
Fluphenazine
Haloperidol
Levomepromazine
Olanzepine
Prochlorperazine
Pericyazine
Perphenazine
Pimozide
Promazine
Quetiapine
Resperidone
Sertindole
Sulpiride
Trifluoperazine
Zotepine
Zuclopenthixol
Anti-hypertensive and other cardiac
Amlodipine
Diltiazem
Enalapril
Lisinopril
Methyldopa
Nifedipine
Nisoldipine
Prazosin
Verapamil
Anti-epileptic drugs
Carbamazine
Valproate acid
Diuretic drugs
Spironolactone
Bumetanide
Anti-depressant drugs
Amitriptyline
H2 receptor antagonist and proton pump inhibitors
Cimetidine
Famotidine
Lasoprazole
Omeprazole
Nizatidine
Ranitidine
Gonadorelin analgues
Buserelin
Goserelin
Leuprorelin
Nafarelin
Tripotorelin
Antibiotic anti-viral and anti-fungal drugs
Atazanavir
Darunavir
Efavirenz
Isoniazid
Ketoconazole
Stavudine
Cytotoxic drugs
Dasatinib
Estramustine
Imatinib
Immunosuppressant drugs
Ciclosporine
Anti-gout drugs
Allopurinol
Hormones
Cyproterone
Ethinylestradiol
Human chorionic gonadrotroophin
Oestrogen
Testosterone
Hormine antagonist
Bicalutaminde
Flutamide
Human menopausal gonadotrophins
Brand names
Menogen – combination drugs: follicle stimulating hormone and leutinising hormone
Menopur
LIST 2
Drugs that can cause gynaecomastia in alphabetical order
Atanazavir
Amlodipine
Allopurinol
Amitriptyline
Aripiorazole
Amisulpiride
Bumetanide
Bicalutamide
Benperiodl
Buserelin
Chorionic Gonadotrophin
Cyproterone
Carbamazepine
Ciclosporine
Chlorpromazine
Clozapine
Cimetidine
Darunavir
Diltiazem
Dasatinib
Digoxin
Dutasteride
Estramustine
Ethinylestradiol
Enalapril
Efavirenz
Famotidine
Flutamide
Flupentixol
Fluphenazine
Finasteride
Goserelin
Haloperidol
Human Chorionic Gonadotrophin
Isoniaxzid
Imatinib
Lanzoprazole
Lisinopril
Leuprorelin
Levomepromazine
Methyldopa
Mitotane
Menogan (brand name)
Menopur (brand name)
Nisoldipine
Nifedipine
Nizatidine
Nafarelin
Oestrogen
Omeprazole
Olanzepine
Prazosin
Prochlorperazine
Pericyazine
Perphenazine
Pimozide
Promazine
Pipothiazine
Quetiapine
Risperidone
Resperidone
Ranitidine
Spironolactone
Stavudine
Sildenafil
Sulpiride
Sertindole
Testosterone and esters
Trifluoperazine
Triptorelin
Verapmil
Zuclopenthixol
Zotepine
Zidovudine
LIST 3
Drugs reported to cause gynaecomastia in isolated case reports.
Atorvastatin
Cetrizine
Clonidine
Fenofibrate
Fluoxetin
Gabapentin
Methotrexate
Paroxetine
Pregabulin
Rofecoxib
Rosuvastatin
Thalidomide
Theophylline
